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142

抑制剂 & 化合物

12

天然产物

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Cat. No. Product Name Target Signaling Pathways
T22260 Aminopurvalanol A

CDK Cell Cycle/Checkpoint
Aminopurvalanol A 是一种竞争性、选择性和细胞渗透性的Cyclins/Cdk 复合物抑制剂,优先靶向G2/M 期转变进而抑制癌细胞分化。它通过抑制生理获能依赖性肌动蛋白聚合而抑制精子受精能力。
T1753 D-64131

Microtubule Associated Cytoskeletal Signaling
D64131 是一种微管蛋白聚合抑制剂,IC50 值为 0.53 μM。它具有抗丝分裂活性,可用于癌症研究。
T19664 ON1231320

GBO-006

Apoptosis; PLK Apoptosis; Cell Cycle/Checkpoint
ON1231320 (GBO-006) 是一种高度特异性的 polo 样激酶 2 抑制剂,IC50为 0.31 µM。在有丝分裂 G2/M 期阻断肿瘤细胞周期进程,它可导致细胞凋亡。它是一种芳基磺酰基吡啶并嘧啶酮,具有抗肿瘤活性。
T3459 VK3-OCH3

2-[(2-Methoxy)ethylthio]-3-methyl-1,4-na

Others Others
VK3-OCH3 (2-[(2-Methoxy)ethylthio]-3-methyl-1,4-na) 是一种通过血红素加氧酶(HO-1) 相关机制的选择性抗肿瘤剂;维生素 K3 类似物。
T10723 CDC25B-IN-1

ethyl 3-[(3-methoxynaphthalen-1-yl)amino]benzoate

Phosphatase Metabolism
CDC25B-IN-1 是 CDC25B 的抑制剂,Ki 为 8.5 μM。 CDC25B-IN-1 通过抑制细胞增殖和集落形成来增加 G2/M 期。
T64923 Sodium citrate

Citrosodine,Natrocitral,柠檬酸钠

Others Others
Sodium citrate (Natrocitral) 是柠檬酸的钠盐。Sodium citrate 诱导G2/M 期和S 期细胞凋亡和细胞周期阻滞。Sodium citrate 通过降低抗氧化酶活性引起肝脏氧化损伤。
T3485 Probimane

AT-2153,MM-159

Others Others
Probimane (AT-2153) 具有抗增殖作用、细胞周期 G2/M 期阻滞和用 MST-16 阻断人类肿瘤细胞系中的染色体分离。
T6864 Ixabepilone

BMS 247550,Ixempra,Azaepothilone B,伊沙匹隆,BMS 247550-1

Apoptosis; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Ixabepilone (Azaepothilone B) 是一种可口服的微管抑制剂,能够与微管蛋白结合,促进微管蛋白的聚合和微管的稳定,使细胞停滞在 G2-M 期,诱导细胞凋亡。
T63732 EGFR-IN-3

Apoptosis; EGFR Angiogenesis; Apoptosis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
EGFR-IN-3 是一种 EGFR 抑制剂,具有潜在的抗肿瘤活性。EGFR-IN-3 抑制 EGFRwt-TK,诱导细胞凋亡 (apoptosis),可使细胞在G2/M期阻滞。
T78701 Tubulin inhibitor 32

Apoptosis Apoptosis
Tubulin inhibitor 32是一种口服活性的新型微管抑制剂,具有抗增殖和抗肿瘤活性,可抑制微管聚合,可诱导细胞凋亡及在G2/M期引起细胞周期停滞。
T67746 IMS2186

Others Others
IMS2186 是一种抗脉络膜新生血管 (CNV) 试剂, 可以使癌细胞周期阻滞在 G2/M 期,由此产生抗增殖和抗血管生成作用。IMS2186 能够减少眼睛渗漏和病变细胞的数量,并且无眼内毒性。
T77729 MY-1076

Apoptosis; YAP Apoptosis; Stem Cells
MY-1076 是一种高效的 YAP 抑制剂,具有抗胃癌活性。MY-1076 剂量依赖性诱导G2/M期阻滞,诱导 YAP 降解和细胞凋亡,抑制微管蛋白聚合。MY-1076 抑制 MGC-803、SGC-7901、HCT-116 和 KYSE450 细胞增殖。
T28886 Suprafenacine

N'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide

Microtubule Associated Cytoskeletal Signaling
Suprafenacine (N'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide) 是一种细胞渗透性微管去稳定剂,可在 G2/M 期诱导细胞周期停滞和细胞凋亡。 它 与微管结合并抑制秋水仙碱连接处的聚集。 它对癌细胞有选择性,包​​括耐药癌细胞。
T63992 KS100

KS100 是 ALDH 的有效抑制剂,能够作用于 ALDH1A1 (IC50: 334 nM)、ALDH2 (IC50: 2137 nM) 和 ALDH3A1 (IC50: 360 nM)。KS100 能够明显提高 ROS 活性、脂质过氧化和有毒醛的积累,且具有低毒性的抗增殖和抗癌活性。KS100 能够将细胞周期阻滞在 G2/M 期,并诱导细胞凋亡 (apoptosis)。
T4451 Estramustine phosphate sodium

Ro 21-8837/001,Estramustine phosphate disodium,雌莫司汀磷酸钠

Apoptosis; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Estramustine phosphate sodium (Ro 21-8837/001) 是雌二醇类似物,是一种具有口服活性抗微管化疗剂,通过与微管相关蛋白和微管蛋白结合而使微管解聚。它可诱导前列腺癌细胞凋亡,可研究前列腺癌。
T77647 Tubulin polymerization-IN-43

Apoptosis; Microtubule Associated Apoptosis; Cytoskeletal Signaling
Tubulin polymerization-IN-43 是一种微管蛋白聚合 (tubulin polymerization) 抑制剂。Tubulin polymerization-IN-43 具有多种作用,通过靶向 Colchicine 位点破坏细胞微管网络,促进白血病细胞的细胞周期停滞在 G2/M 期和细胞凋亡 (apoptosis)。Tubulin polymerization-IN-43 具有抗血管生成活性。
T2090 Lexibulin

CYT-997

Apoptosis; Reactive Oxygen Species; Microtubule Associated Apoptosis; Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB
Lexibulin (CYT-997) 是一种微管蛋白聚集强效抑制剂,可诱导细胞凋亡,并诱导 GC 细胞中的线粒体ROS 生成。它对多种癌细胞的 IC50 值为 10-100n M,在体内外具有高细胞毒性和血管增生阻断作用。
T3124 Carbendazim

Bavistin,Carbendazole,多菌灵,Mercarzole

Antifungal Microbiology/Virology
Carbendazim (Mercarzole) 是一种具有抗肿瘤活性的苯并咪唑衍生物,可用于癌症研究。它是一种口服广谱苯并咪唑杀菌剂,可作为真菌疾病研究的杀虫剂。
T41163 ZNL 02-096

Pomalidomide-C3-adavosertib

Apoptosis; Wee1 Apoptosis; Cell Cycle/Checkpoint
ZNL 02-096 (Pomalidomide-C3-adavosertib) 是一种快速和选择性的 Wee1 降解剂 (IC50=3.58 nM)。ZNL 02-096 可在亚摩尔浓度下选择性降解 Wee1,而不损伤 AZD 1775 的二级靶点 PLK1。在体外 MOLT-4 细胞中,ZNL 02-096 可诱导 Wee1 降解、DNA 损伤积累、细胞周期停滞在 G2/M 期和细胞凋亡。ZNL 02-096 在 300 种癌症细胞系中显示出抗增殖作用。
T13901 SS28

Microtubule Associated Cytoskeletal Signaling
SS28 inhibits tubulin polymerization to cause cell cycle arrest at G2/M phase.
T31004 Compound 8H

Compound-8H,Compound 8-H,Compound 343

Compound 8H is an inducer of G2/M-phase cell cycle arrest and cell death in cancer cell lines.
T30768 CB-403

UNII-4V9Q0C88UK,CB403,CB 403

CB-403 is a cinnamaldehyde derivative that has antitumor effects by blocking cell cycle progression in the G2/M phase.
T13227 Tubulin inhibitor 1

Microtubule Associated Cytoskeletal Signaling
Tubulin inhibitor 1 is an inhibitor of tubulin, inhibits tubulin polymerization, with potent anti-tumor activity, induces cellular apoptosis causes and cellular mitotic arrest in the G2/M phase.
T62458 EGFR-IN-56

EGFR-IN-56 (Compound 13a) 是一种 EGFR 的有效抑制剂,能够作用于 EGFRT790M (IC50: 541.7 nM) 和 EGFRT790M/L858R (IC50: 132.1 nM)。EGFR-IN-56 能够将癌细胞的细胞周期阻滞在 G2/M 期,并诱导细胞凋亡 (apoptosis)。
T83020 Antiproliferative agent-37

Antiproliferative agent-37 (compound 10J) 通过诱导细胞周期在G2/M期的阻滞来实现其抗增殖效果。
T23817 BPTQ

B-P-T-Q

BPTQ is a typical intercalator of DNA that acts by inducing a dose-dependent inhibitory effect on the proliferation of cancer cells by arresting cells at the S and G2/M phase.
T61129 Tubulin polymerization-IN-27

Tubulin polymerization-IN-27 (compound 5j) is an inhibitor of tubulin polymerization. It has the ability to halt the cell cycle specifically at the G2/M phase and also induce apoptosis [1].
T73413 Cadein1

Cadein1 是一种异喹啉衍生物,在p53功能缺失的癌细胞中,可导致 G2/M 延迟和caspase 依赖的凋亡。
T79463 Antitumor agent-110

Apoptosis Apoptosis
Antitumor agent-110 (compound 13) 是一种抗癌咪唑四嗪,具备良好的渗透性,能够阻滞细胞周期于G2/M期并诱导apoptosis。
T61401 3-(3-Phenoxybenzyl)amino-β-carboline

3-(3-Phenoxybenzyl)amino-β-carboline is a highly effective tubulin inhibitor, selectively degrading αβ-tubulin heterodimers. It induces cell cycle arrest and apoptosis in the G2/M phase. Additionally, 3-(3-Phenoxybenzyl)amino-β-carboline displays notable anticancer activity [1].
T61616 Antitumor agent-38

Antitumor agent-38 is a highly effective antitumor compound that exhibits antiproliferative activity towards cancer cells. It induces cell cycle arrest specifically at the late S and G2/M phase, while not impeding microtubule formation or altering cell morphology [1].
T36700 CKD 602

Topoisomerase I inhibitor. Forms stable DNA-topoisomerase complexes during DNA replication and induces cell cycle arrest in the G2/M phase. Inhibits growth of a range of cancer cell lines in vitro, as well as of ovarian and leukemia tumors in vivo.
T61779 STAT3-IN-9

STAT3-IN-9, a potent inhibitor of STAT3 activation at Tyr705, exhibits no impact on the phosphorylation of STAT1 at Tyr 701. Additionally, this compound efficiently induces apoptosis and cell cycle arrest specifically at the G2/M phase [1].
T63271 Antitumor agent-62

Antitumor agent-62 是释放 NO 的抗肿瘤剂,对癌细胞表现出抗增殖作用,能够激活线粒体凋亡 (apoptosis) 通路,能够将细胞周期阻滞到 G2/M 期。
T60505 Antitumor agent-43

Antitumor agent-43 (Compound 4B) 是一种有效的抗肿瘤剂,可诱导细胞周期阻滞在G2/M 期。Antitumor agent-43对 T-24 细胞的IC50值为0.5 μM。
T63304 Topoisomerase II inhibitor 9

Topoisomerase II inhibitor 9 是 Topo II 抑制剂 (IC50: 0.97 μM),也是 DNA 嵌入剂 (IC50: 43.51 μM),能够在 G2/M 期阻滞 Hep G‐2 细胞周期,诱导细胞凋亡 (apoptosis)。
T68570 TPI-287

TPI 287 is a synthetic, third generation taxane with potential antineoplastic activity. TPI 287 binds to tubulin and stabilizes microtubules, resulting in inhibition of microtubule assembly/disassembly dynamics, cell cycle arrest at the G2/M phase, and apoptosis.
T62796 VEGFR-2-IN-13

VEGFR-2-IN-13 (Compound 19a) 是一种有效的 VEGFR-2 抑制剂 (IC50: 3.4 nM)。VEGFR-2-IN-13 能够将 HepG2 的细胞周期停滞在 G2/M 期,诱导细胞凋亡 (apoptosis)。
T79429 Tubulin polymerization-IN-50

Tubulin polymerization-IN-50(compound 7n)是一种Tubulin polymerization抑制剂,其在SK-Mel-28细胞中的IC50值为5.05 μM,能够诱导(cell cycle)阻滞在G2/M期。
T62693 Tubulin polymerization-IN-29

Tubulin polymerization-IN-29 是一种有效的微管蛋白聚合抑制剂,显示出有效的抗增殖效果。Tubulin polymerization-IN-29 能够诱导 HeLa 细胞的细胞周期阻滞在 G2/M 期。
T78686 Apoptosis inducer 11

Apoptosis Apoptosis
Apoptosisinducer 11(compound 3u)通过线粒体途径引发细胞凋亡。在非霍奇金淋巴瘤细胞系中,该化合物导致G2/M期停滞和S期显著减少。
T60735 Tubulin polymerization-IN-22

Tubulin aggregation-IN-22 抑制细胞周期在 G2/M 期,并且诱导细胞凋亡。Tubulin aggregation-IN-22 是一种微管蛋白聚合抑制剂 (IC50 = 8.1 μM)。
T72205 Antiproliferative agent-19

Antiproliferative agent-19 (化合物 4a) 作为一种抗癌剂,通过诱导细胞凋亡和细胞周期在G2/M期的停滞来对肺癌细胞展现抗增殖活性。
T60452 PCAF-IN-2

PCAF-IN-2 (compound 17) 是一种有效的 PCAF 抑制剂(IC50 = 5.31 µM)。PCAF-IN-2 具有抗肿瘤活性。PCAF-IN-2 诱导细胞凋亡并且阻滞细胞周期在 G2/M 期。
T60776 Anticancer agent 68

Anticancer agent 68 is (Compound 12) 是一种抗癌剂。Anticancer agent 68 将细胞阻滞在 G2/M 期并诱导程序性细胞死亡。Anticancer agent 68 通过激活 p53 和 PTEN 诱导上调肿瘤抑制。
T60766 Topoisomerase I inhibitor 3

Topoisomerase I inhibitor 3 (Compound ZML-14) 诱导 HepG2 细胞凋亡,并在 G2/M 期阻滞细胞周期。Topoisomerase I inhibitor 3 是与拓扑异构酶 I-DNA 复合物相互作用的拓扑异构酶 I 抑制剂。
T60781 Topoisomerase II inhibitor 8

Topoisomerase II inhibitor 8 (化合物 22) 显示出良好的抗增殖活性,并将细胞周期阻滞在 G2/M 期。Topoisomerase II inhibitor 8是拓扑异构酶 II 的有效抑制剂 (IC 50 = 0.52 μM)。
T78862 EGFR-IN-86

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
EGFR-IN-86(化合物4i)是一种高效的EGFR抑制剂,IC50为1.5 nM,对胶质母细胞瘤表现出强抗癌活性。该化合物能够诱导细胞凋亡并使U87细胞周期在G2/M期发生阻滞。
T69316 DA 3003-2

NSC663285

DA 3003-2为一种高效的选择性Cdc25抑制剂,展示了抗增殖活性,能诱导细胞周期在G2/M期停滞,并提高P-tyr15Cdc2表达量,显示出对前列腺癌研究的应用潜力。
T78940 EGFR-IN-78

Apoptosis Apoptosis
EGFR-IN-78(compound A5)为2-氨基嘧啶衍生物,既是EGFRC797S-TK的可逆抑制剂,也能诱导细胞凋亡(apoptosis)。该化合物展现抗增殖能力,阻止EGFR磷酸化,导致细胞周期在G2/M期暂停。

化合物

Aminopurvalanol A
Cat.No: T22260
Synonym:
Target: CDK
D-64131
Cat.No: T1753
Synonym:
Target: Microtubule Associated
ON1231320
Cat.No: T19664
Synonym: GBO-006
Target: Apoptosis, PLK
VK3-OCH3
Cat.No: T3459
Synonym: 2-[(2-Methoxy)ethylthio]-3-methyl-1,4-na
Target: Others
CDC25B-IN-1
Cat.No: T10723
Synonym: ethyl 3-[(3-methoxynaphthalen-1-yl)amino]benzoate
Target: Phosphatase
Sodium citrate
Cat.No: T64923
Synonym: Citrosodine,Natrocitral,柠檬酸钠
Target: Others
Probimane
Cat.No: T3485
Synonym: AT-2153,MM-159
Target: Others
Ixabepilone
Cat.No: T6864
Synonym: BMS 247550,Ixempra,Azaepothilone B,伊沙匹隆,BMS 247550-1
Target: Apoptosis, Microtubule Associated
EGFR-IN-3
Cat.No: T63732
Synonym:
Target: Apoptosis, EGFR
Tubulin inhibitor 32
Cat.No: T78701
Synonym:
Target: Apoptosis
IMS2186
Cat.No: T67746
Synonym:
Target: Others
MY-1076
Cat.No: T77729
Synonym:
Target: Apoptosis, YAP
Suprafenacine
Cat.No: T28886
Synonym: N'-[(E)-(4-methylphenyl)methylidene]-4,5,6,7-tetrahydro-1H-indazole-3-carbohydrazide
Target: Microtubule Associated
KS100
Cat.No: T63992
Synonym:
Target:
Estramustine phosphate sodium
Cat.No: T4451
Synonym: Ro 21-8837/001,Estramustine phosphate disodium,雌莫司汀磷酸钠
Target: Apoptosis, Microtubule Associated
Tubulin polymerization-IN-43
Cat.No: T77647
Synonym:
Target: Apoptosis, Microtubule Associated
Lexibulin
Cat.No: T2090
Synonym: CYT-997
Target: Apoptosis, Reactive Oxygen Species, Microtubule Associated
Carbendazim
Cat.No: T3124
Synonym: Bavistin,Carbendazole,多菌灵,Mercarzole
Target: Antifungal
ZNL 02-096
Cat.No: T41163
Synonym: Pomalidomide-C3-adavosertib
Target: Apoptosis, Wee1
SS28
Cat.No: T13901
Synonym:
Target: Microtubule Associated
Compound 8H
Cat.No: T31004
Synonym: Compound-8H,Compound 8-H,Compound 343
Target:
CB-403
Cat.No: T30768
Synonym: UNII-4V9Q0C88UK,CB403,CB 403
Target:
Tubulin inhibitor 1
Cat.No: T13227
Synonym:
Target: Microtubule Associated
EGFR-IN-56
Cat.No: T62458
Synonym:
Target:
Antiproliferative agent-37
Cat.No: T83020
Synonym:
Target:
BPTQ
Cat.No: T23817
Synonym: B-P-T-Q
Target:
Tubulin polymerization-IN-27
Cat.No: T61129
Synonym:
Target:
Cadein1
Cat.No: T73413
Synonym:
Target:
Antitumor agent-110
Cat.No: T79463
Synonym:
Target: Apoptosis
3-(3-Phenoxybenzyl)amino-β-carboline
Cat.No: T61401
Synonym:
Target:
Antitumor agent-38
Cat.No: T61616
Synonym:
Target:
CKD 602
Cat.No: T36700
Synonym:
Target:
STAT3-IN-9
Cat.No: T61779
Synonym:
Target:
Antitumor agent-62
Cat.No: T63271
Synonym:
Target:
Antitumor agent-43
Cat.No: T60505
Synonym:
Target:
Topoisomerase II inhibitor 9
Cat.No: T63304
Synonym:
Target:
TPI-287
Cat.No: T68570
Synonym:
Target:
VEGFR-2-IN-13
Cat.No: T62796
Synonym:
Target:
Tubulin polymerization-IN-50
Cat.No: T79429
Synonym:
Target:
Tubulin polymerization-IN-29
Cat.No: T62693
Synonym:
Target:
Apoptosis inducer 11
Cat.No: T78686
Synonym:
Target: Apoptosis
Tubulin polymerization-IN-22
Cat.No: T60735
Synonym:
Target:
Antiproliferative agent-19
Cat.No: T72205
Synonym:
Target:
PCAF-IN-2
Cat.No: T60452
Synonym:
Target:
Anticancer agent 68
Cat.No: T60776
Synonym:
Target:
Topoisomerase I inhibitor 3
Cat.No: T60766
Synonym:
Target:
Topoisomerase II inhibitor 8
Cat.No: T60781
Synonym:
Target:
EGFR-IN-86
Cat.No: T78862
Synonym:
Target: EGFR
DA 3003-2
Cat.No: T69316
Synonym: NSC663285
Target:
EGFR-IN-78
Cat.No: T78940
Synonym:
Target: Apoptosis
Cat. No. Product Name Target Signaling Pathways
TQ0089 Juglanin

Apoptosis; JNK; Autophagy Apoptosis; Autophagy; MAPK
Juglanin 是来自金鸡脚的一种黄酮类天然产物,是一种 JNK 的激活剂,能诱导人乳腺癌细胞的凋亡和自噬,具有炎症和抗肿瘤活性。
T5669 Citric acid monohydrate

Others Others
Citric acid monohydrate 是一种存在于柑橘类水果中的三羧酸。柠檬酸因其抗氧化特性而被用作药物制剂中的赋形剂。它保持活性成分的稳定性并用作防腐剂。
T5S0636 Citric acid

柠檬酸,Citro,Citretten

Apoptosis; Others; Endogenous Metabolite; Antibacterial; Antibiotic Apoptosis; Metabolism; Microbiology/Virology; Others
Citric acid (Citro) 是柑橘类水果中发现的弱有机三羧酸。柠檬酸是食品添加剂和天然防腐剂。
TN2058 Persicogenin

Anti-infection Microbiology/Virology
Persicogenin 是分离自 Rhus retinorrhoea 中,具有抗癌作用。
T4S1335 Daphnoretin

Dephnoretin,西瑞香素,Thymelol

Influenza Virus; Caspase; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome
Daphnoretin (Thymelol) 是从了哥王中提取得到的一种天然产物,具有抗癌和抗病毒活性。它通过在 G2/M 期连续阻断细胞并激活 caspase-3 通路导致 HOS 细胞死亡。
T81818 Metachromins X

Metachromins X,一倍半萜醌类化合物,能阻碍HeLa/Fucci2细胞在S/G2/M期的细胞周期。
TN5190 Tryprostatin A

Topoisomerase; Antifection DNA Damage/DNA Repair; Microbiology/Virology
Tryprostatin A is an inhibitor of breast cancer resistance protein. Tryprostatin A and tryprostatin B are indole alkaloid-based fungal products that inhibit mammalian cell cycle at the G2/M phase.
TN5336 9-Oxo-10,11-dehydroageraphorone

4,7(11)-Cadinadiene-3,8-dione,DTD,7,11-Dehydro-8-oxoageraphorone,泽兰二酮

9-Oxo-10,11-dehydroageraphorone has acaricidal activity. It induces hepatotoxicity and cholestasis in rats. 9-Oxo-10,11-dehydroageraphorone also effectively inhibits the proliferation of HeLa cells by arresting the cell cycle transition from S to G2/M pha
TN2344 Swainsonine

Tridolgosir

Apoptosis; Others; Antibiotic Apoptosis; Microbiology/Virology; Others
Swainsonine (Tridolgosir) 是一种从黄芪中分离出来的一种生物碱,是一种强效和可逆的α-甘露糖苷酶抑制剂。Swainsonine 具有抗肿瘤活性,可诱导细胞凋亡和细胞周期停滞在 G2/M 期。
T75602 Albanol B

Albanol B 是一种芳基苯并呋喃衍生物,可从桑葚中分离得到。Albanol B 具有抗阿尔茨海默病、抗菌和抗氧化活性。Albanol B 抑制癌细胞增殖,下调 CDK1表达。Albanol B 还会诱导细胞周期停滞在 G2/M 期,诱导细胞凋亡 (apoptosis)。Albanol B 诱导线粒体 ROS 产生并增加 AKT 和 ERK1/2的磷酸化水平。
T36961 Malformin C

Malformin C is a natural fungus-derived bicyclic pentapeptide that has antibacterial properties, particularly against species of Bacillus. Malformin C potently blocks the ability of bleomycin to induce G2 arrest in human T-cell leukemia-derived Jurkat cells (IC50 = 0.9 nM). It less potently abrogates colchicine-induced M phase arrest in Jurkat cells (IC50 = 24 nM). Malformin C inhibits cell growth dose-dependently in Colon 38 and HCT 115 cancer cells (IC50s = 0.27 and 0.18 μM, respectively) but ...
TN5639 Rocaglaol

Ferrugin,Aglaiastatin A

Rocaglaol is a potent anticancer drug that induces apoptosis of LNCaP cells through the mitochondrial pathway and its G2/M-phase cell cycle arrest is associated with the down-regulation of Cdc25C and the dephosphorylation of Cdc2. Rocaglaol can reduce tis

天然产物

Juglanin
Cat.No: TQ0089
Synonym:
Target: Apoptosis, JNK, Autophagy
Citric acid monohydrate
Cat.No: T5669
Synonym:
Target: Others
Citric acid
Cat.No: T5S0636
Synonym: 柠檬酸,Citro,Citretten
Target: Apoptosis, Others, Endogenous Metabolite, Antibacterial, Antibiotic
Persicogenin
Cat.No: TN2058
Synonym:
Target: Anti-infection
Daphnoretin
Cat.No: T4S1335
Synonym: Dephnoretin,西瑞香素,Thymelol
Target: Influenza Virus, Caspase, PKC
Metachromins X
Cat.No: T81818
Synonym:
Target:
Tryprostatin A
Cat.No: TN5190
Synonym:
Target: Topoisomerase, Antifection
9-Oxo-10,11-dehydroageraphorone
Cat.No: TN5336
Synonym: 4,7(11)-Cadinadiene-3,8-dione,DTD,7,11-Dehydro-8-oxoageraphorone,泽兰二酮
Target:
Swainsonine
Cat.No: TN2344
Synonym: Tridolgosir
Target: Apoptosis, Others, Antibiotic
Albanol B
Cat.No: T75602
Synonym:
Target:
Malformin C
Cat.No: T36961
Synonym:
Target:
Rocaglaol
Cat.No: TN5639
Synonym: Ferrugin,Aglaiastatin A
Target:
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